Cinacalcet Hydrochloride + Flecainide Interaction

Majorinteraction on record

Description

Cinacalcet is a strong CYP2D6 inhibitor. Dose adjustments may be required, particularly for drugs with narrow therapeutic index such as flecainide.

Mechanism

Cinacalcet inhibits CYP2D6 metabolism of flecainide

Source: NLP:cinacalcet hydrochloride