Cimetidine + Pioglitazole And Metformin Hydrochloride Interaction

Majorinteraction on record

Description

Reduces metformin clearance, increasing systemic exposure and risk for lactic acidosis. Consider benefits and risks of concomitant use.

Mechanism

Inhibits renal tubular transport of metformin (OCT2/MATE)

Source: NLP:pioglitazone hydrochloride and metformin hydrochloride