Cholic Acid + Cyclosporine Interaction
Majorinteraction on record
Description
BSEP inhibitor that may exacerbate accumulation of conjugated bile salts in liver. Avoid concomitant use; if necessary, monitor serum transaminases and bilirubin.
Mechanism
Inhibition of bile salt efflux pump (BSEP) increases hepatic bile salt accumulation
Source: NLP:cholic acid