Bictegravir Sodium Emtricitabine And Tenofovir Alafenamide F + Dofetilide Interaction
Moderateinteraction on record
Description
BIC inhibits OCT2 and MATE1, which may increase dofetilide plasma concentrations.
Mechanism
Inhibition of organic cation transporter 2 (OCT2) and multidrug and toxin extrusion transporter 1 (MATE1)
Source: NLP:bictegravir sodium, emtricitabine, and tenofovir alafenamide fumarate