Bexarotene + Paclitaxel Interaction

Moderateinteraction on record

Description

Bexarotene decreased paclitaxel exposure (AUC) by 19%. When combined with carboplatin, paclitaxel exposure was increased 2-fold.

Mechanism

CYP3A4 and CYP2C8 induction by bexarotene

Source: NLP:bexarotene