Belumosudil + P Gp Or Bcrp Substrates Interaction
Majorinteraction on record
Description
Belumosudil affects P-gp substrates for which minimal concentration changes may lead to serious toxicities. Avoid concomitant use where possible; if necessary, decrease substrate dosages.
Mechanism
Belumosudil is a P-gp inhibitor
Source: NLP:belumosudil