Azelastine Hydrochloride Fluticasone Propionate + Ritonavir Interaction
Contraindicatedinteraction on record
Description
Strong CYP3A4 inhibitor that significantly increases fluticasone propionate plasma exposure and reduces serum cortisol, resulting in systemic corticosteroid effects including Cushing syndrome and adrenal suppression.
Mechanism
CYP3A4 inhibition
Source: NLP:azelastine hydrochloride and fluticasone propionate