Azelastine Hydrochloride Fluticasone Propionate + Ketoconazole Interaction
Majorinteraction on record
Description
Strong CYP3A4 inhibitor that increases fluticasone propionate plasma exposure and reduces cortisol AUC. Caution should be exercised when coadministered.
Mechanism
CYP3A4 inhibition
Source: NLP:azelastine hydrochloride and fluticasone propionate