Atrasentan + Gemfibrozil Interaction
Moderateinteraction on record
Description
OATP1B1 substrate; gemfibrozil inhibition may increase atrasentan exposure, requiring dosing reduction.
Mechanism
OATP1B1 transporter inhibition
Source: NLP:gemfibrozil
OATP1B1 substrate; gemfibrozil inhibition may increase atrasentan exposure, requiring dosing reduction.
OATP1B1 transporter inhibition
Source: NLP:gemfibrozil