Atogepant + Rifampin Interaction

Moderateinteraction on record

Description

Strong CYP3A4 inducer and OATP1B1/OATP1B3 inhibitor resulting in significant decrease in atogepant exposure; dosage adjustment and monitoring for reduced efficacy recommended.

Mechanism

CYP3A4 induction and OATP inhibition

Source: NLP:atogepant