Artemether And Lumefantrine + Rifampin Interaction
Contraindicatedinteraction on record
Description
Strong CYP3A4 inducer causing significant decreases in artemether (89%), DHA (85%), and lumefantrine (68%) exposure, resulting in loss of antimalarial efficacy.
Mechanism
CYP3A4 induction
Source: NLP:artemether and lumefantrine