Amiodarone Hydrochloride + Lidocaine Interaction

Moderateinteraction on record

Description

CYP3A substrate. Sinus bradycardia reported with oral amiodarone and lidocaine for local anesthesia. Monitor heart rate; lower starting dose may be required.

Mechanism

CYP3A inhibition and pharmacodynamic interaction

Source: NLP:amiodarone hydrochloride