Ado Trastuzumab Emtansine + Nefazodone Interaction

Majorinteraction on record

Description

Strong CYP3A4 inhibitor that may increase DM1 exposure and toxicity. Concomitant use should be avoided or KADCYLA treatment delayed.

Mechanism

Inhibition of CYP3A4-mediated metabolism of DM1

Source: NLP:ado-trastuzumab emtansine