Cobimetinib + Itraconazole Interaction
Moderateinteraction on record
Description
( 2.3 , 7.1 , 7.2 ) 7.1 Effect of Strong or Moderate CYP3A Inhibitors on COTELLIC Coadministration of COTELLIC with itraconazole (a strong CYP3A4 inhibitor) increased cobimetinib systemic exposure by 6.7-fold.
Source: FDA drug label - cobimetinib