Abemaciclib + Ketoconazole Interaction
Majorinteraction on record
Description
7 DRUG INTERACTIONS CYP3A Inhibitors: Avoid concomitant use of ketoconazole. Ketoconazole Avoid concomitant use of ketoconazole. Ketoconazole is predicted to increase the AUC of abemaciclib by up to 16-fold [see Clinical Pharmacology ( 12.3 )] .
Source: FDA drug label - abemaciclib